BOLD-100 with FOLFOX for Advanced Gastrointestinal Cancers

This study is testing BOLD-100, a new drug, in combination with standard FOLFOX chemotherapy for advanced gastrointestinal cancers like colorectal, pancreatic, gastric cancers, and cholangiocarcinoma. BOLD-100 works by decreasing a protein called GRP78 in cancer cells. The study aims to find the safest and most effective dose of BOLD-100 when given with FOLFOX. You might be able to join if you are 18 or older and have certain types of advanced gastrointestinal tumors. For colorectal cancer, you must have had only one prior treatment for metastatic disease and not received oxaliplatin. The main goals are to track any side effects and how well the treatment is tolerated. Enrollment in some parts of the study (Arms I-VI) is closed, but Arm VII, specifically for colorectal cancer, is still enrolling participants.

Study design
This is a multi-center, non-randomized study, but Arm VII for colorectal cancer will randomize participants to receive one of two doses of BOLD-100 plus FOLFOX, or FOLFOX alone, in a 1:1:1 ratio. The study plans to enroll 220 participants.
What's involved
Participants will receive BOLD-100 combined with FOLFOX chemotherapy. You will undergo physical exams, ECGs (heart tests), vital sign checks, and lab tests throughout the study and for about two weeks after your last treatment.
Compensation
Not stated in the trial record.
Follow-up
You will be followed through study completion, which is approximately two weeks after your last treatment, to monitor for side effects and other health changes.

AI-generated from the public study record. Only the study team can confirm whether you're eligible — confirm details with them before making decisions.

NCT04421820

BOLD-100 in Combination With FOLFOX for the Treatment of Advanced Solid Tumours

Recruiting
PHASE1Ages 18+InterventionalTreatment
Bold Therapeutics, Inc.
~220 participants
Updated 2026-05-18 on ClinicalTrials.gov
What's tested:BOLD-100 +/- FOLFOX Chemotherapy (Arm VII)BOLD-100 in combination with FOLFOX Chemotherapy (Arms I-VI)

At a glance

Recruiting sites
16 of 24 listed sites are recruiting right now
RecruitingSuspended, closed, or not yet open
What they're measuring
Incidence and severity of adverse events ([S]AEs)
Measured over Through study completion, approximately 2 weeks after last treatment
+5 more outcomes measured
Colorectal Cancer
Pancreatic Cancer
Gastric Cancers
Cholangiocarcinoma
24 sites across 10 states
South Korea5
Ontario3
Ireland3
Italy3
Spain3
Quebec2
Germany2
California1

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  • Incidence and severity of adverse events ([S]AEs)Through study completion, approximately 2 weeks after last treatment

    Arms I-VI: Primary outcome measure; Arm VII: Secondary outcome measure

  • Incidence of dose-limiting toxicities (DLT)Screening to 4 weeks after first treatment

    Dose escalation only.

  • Incidence of clinically significant changes or abnormalities from Physical Examinations, ECGs, Vital Signs, Laboratory Results, ECOG performance statusThrough study completion, approximately 2 weeks after last treatment

    Arms I-VI: Primary outcome measure; Arm VII: Secondary outcome measure

  • Progression Free Survival (PFS): Arm VIIThrough study completion, approximately 2 weeks after last treatment for last patient

    Arm VII: Primary outcome measure

  • Overall Response Rate (ORR): Arm VIIThrough study completion, approximately 2 weeks after last treatment for last patient

    Arm VII: Primary outcome measure

  • Overall Survival (OS): Arm VIIThrough study completion, approximately 2 weeks after last treatment for last patient

    Arm VII: Primary outcome measure