GNS561 and Trametinib for Advanced KRAS-Mutated Cholangiocarcinoma

This study is testing a combination of two drugs, GNS561 and trametinib, for patients with advanced cholangiocarcinoma (bile duct cancer) that has a specific genetic change called a KRAS mutation. You might be able to join if your cancer has progressed after standard chemotherapy and you have a KRAS mutation. Researchers want to see how safe the drug combination is and how well it shrinks tumors. The study is currently recruiting about 98 participants.

Study design
This is an open-label, multi-center Phase 1b/2a study, meaning both you and your doctors will know which drugs you are receiving. It aims to enroll about 98 participants.
What's involved
Not specified in the trial record.
Compensation
Not stated in the trial record.
Follow-up
The study will measure how well the treatment works for up to 11 months.

AI-generated from the public study record. Only the study team can confirm whether you're eligible — confirm details with them before making decisions.

NCT05874414

Combination of GNS561 and Trametinib in Patients With Advanced KRAS Mutated Cholangiocarcinoma

Recruiting
PHASE1Ages 18+InterventionalTreatment
Genfit
~98 participants
Updated 2026-07-13 on ClinicalTrials.gov
What's tested:GNS561 + Trametinib

At a glance

Recruiting sites
9 of 11 listed sites are recruiting right now
RecruitingSuspended, closed, or not yet open
What they're measuring
Incidence of dose limiting toxicity (DLT) of GNS561 with trametinib (Phase 1b)
Measured over At the end of Cycle 1 (each Cycle is 21 days)
+1 more outcome measured
Cholangiocarcinoma
11 sites across 9 states
California2
Florida2
Illinois1
New York1
Pennsylvania1
Texas1
Virginia1
Wisconsin1
  • Pejvack MOTLAGH, CMO · STUDY_DIRECTOR · Genfit

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  • Incidence of dose limiting toxicity (DLT) of GNS561 with trametinib (Phase 1b)At the end of Cycle 1 (each Cycle is 21 days)

    Defined as Treatment Emergent Adverse Event (TEAE) being at least possibly related to study drug: With Grade ≥ 3 (using NCI CTCAE Version 5.0 or higher as applicable) such as specified in the protocol

  • Objective response rate (ORR) of the combination of GNS561 with trametinib (Phase 2a)Up to 11 months (estimated)

    Defined as the proportion of patients with a best overall response of complete response (CR) or partial response (PR) using Response Evaluation Criteria in Solid Tumors version 1.1 (RECIST v1.1)